Inoa | N- (n- (n-glycylglycycycycycycycycycyl) glycyl) -8-l-l-l-litsineinsin |
Ka helu helu | 14636-12-5 |
Mlecular noncula | C52h74nm dedhot |
Kaupaona molebular | 1227.37 |
Nā helu einecs | 238-680-8-8 |
Makaʻikua | 1824.0 ± 65.0 ° C (wānanaʻia) |
Huakai | 1.46 ± 0.1 g / cm3 (wānana) |
Nā kūlana mālama | E hoʻomau i ka wahiʻeleʻele, i loko o ka lewa i loko o ka lewa, kūʻai aku ma freezer, ma lalo o -15 |
Acidity chee | (PKA) 9.90 ± 0.15 (wānanaʻia) |
[N-α-triglycycyl-8-lysine]-70: pn: wn: wo2010033207sequ 1-triglycyl-8-lysinevasopsin; Nα-glycyl-glycyl-glycyl- [8-lysine] -vasopressi; Nα-glycyl-glycyl-mysine-vasopressin; Nα-glycycycycycycycycycycycycycycycycycyl-vasopressin; Nα-gly-gly-gly-gly-bly-vasopressin; ʻO Terlipressini,ʻo Terlipresse,ʻo TerilipressI, Terlipressinu, Terlipressium.
ʻO Terlipressin,ʻo ia ka inoa o ka inoaʻo kemika ma keʻano he vasopressin maropressin Heʻano prdrug,ʻo ia ka mea i loaʻaʻole iā ia iho. Ua hanaʻia e Aminopeptidase i Vivo e lohi i ka "hoʻokuʻu" i ka hanaʻo LYSINE RASINE ma hope o ka laweʻana i nā nohona oʻekolu ma o kona mau haleʻekolu. No laila, hanaʻo Strlipressin e like me ka mea nāna e hoʻoponopono i ka mea nāna e hoʻopiʻi i ka lysine vasopressin ma ka manawa paʻa.
ʻO ka hopena pharmacocorical o Terlipressin ka mea e hoʻopili ai i ka mika slipcular vascular a hōʻemi i ke kahe koko. Ma nāʻaoʻao'ē aʻe, hiki iā ia ke hōʻemi i ka koloniʻana o ka hoʻopiliʻana, hoʻomaikaʻiʻana i ka hana kōkua ma ka maʻi hepatorenal. ʻO Terlipressin keʻano o ka lāʻau lapaʻau e hiki ke hoʻomaikaʻi i ke ola ola o nā mea maʻi me nā mea maʻi esophagel. Ua hoʻohana nuiʻia ia ma ka mālama ponoʻana i ka lāʻau hemorrhage. Eia kekahi, ua hoʻohana maikaʻiʻiaʻo Terlipressin i ka hana a me ke keiki kāne. Ma ka laulā, e pāʻani paha ia i kahi hana maikaʻi ma keʻano o ka chextory chextoring check a me cardiopulmonary resuscitation resuscitation. Ua hoʻohālikelikeʻia me Vasopressin, he hopena lōʻihi loa ia,ʻaʻole ia e hana i nā hoʻopiʻi maikaʻi loa a me nā hoʻopiʻi koʻikoʻi. Hoʻopakele a me ka mālamaʻana i nā maʻi maʻi maʻi.