,
Inoa | Paclitaxel |
Helu CAS | 33069-62-4 |
ʻAno molekala | C47H51NO14 |
Kaumaha molekula | 853.92 |
Helu EINECS | 608-826-9 |
Lae paila | 774.66°C(Wanamua) |
ʻO ka mānoanoa | 0.200 |
Kūlana mālama | Hoʻopaʻa ʻia i kahi maloʻo, E mālama i loko o ka pahu hau, 2-8 ° C |
Puka | Pauda |
kalakala | Keʻokeʻo |
Hoʻopili | ʻeke PE + ʻeke Aluminum |
Paclitaxel HCL;Paclitaxel(maoli maoli);Paclitaxelx;N-BENZYL-BETA-PHENYLISOSERINE ESTER;PACLITAXEL, TAXUS BREVIFOLIA;PACLITAXEL, TAXUS SPECIES;PACLITAXOL;PACLITAXEL
wehewehe
ʻO Paclitaxel kahi monomeric diterpenoid i unuhi ʻia mai ka ʻili o ka lāʻau maoli ʻo Taxus lāʻau.Ua hōʻike ʻia ka ʻimi ʻana i ka isotope e pili wale ana ka paclitaxel i nā microtubules polymerized a ʻaʻole i pane me nā dimer tubulin unpolymerized.Ma hope o ka ʻike ʻia ʻana o nā cell i ka paclitaxel, e hōʻiliʻili ʻia ka nui o nā microtubules i loko o nā pūnaewele.ʻO ka hōʻiliʻili ʻana o kēia mau microtubules e hoʻopilikia i nā hana like ʻole o nā cell, ʻoi aku ka paʻa o ka māhele cell i ka mitotic phase a poloka i ka mahele maʻamau o nā cell.Ma o Ⅱ-Ⅲ noiʻi lapaʻau, kūpono ka paclitaxel no ka maʻi maʻi ovarian a me ka maʻi kanesa o ka umauma, a loaʻa pū kekahi hopena curative i ka maʻi kanesa, colorectal cancer, melanoma, poʻo a me ka ʻāʻī maʻi, lymphoma a me ka lolo lolo.
Nā hōʻailona
He hopena maikaʻi ia i ka mālama ʻana i ka maʻi maʻi ovarian a me ka platinum a me nā maʻi maʻi ovarian refractory a me ka maʻi maʻi umauma.ʻO ka maʻi maʻi, ka maʻi maʻi ʻōpū o luna, ka maʻi maʻi ʻaʻai liʻiliʻi a me ka maʻi ʻaʻaʻa ʻole liʻiliʻi he manaʻo maikaʻi.
Hoʻohana
E hoʻohana i ka 1: Nā hua lāʻau anti-tumor ākea ākea no ka maʻi maʻi ovarian, ka maʻi maʻi umauma, etc.
E hoʻohana i ka 2: nā lāʻau lapaʻau anti-tumor ākea ākea no ka mālama ʻana i ka maʻi maʻi ovarian, ka maʻi maʻi umauma a me nā maʻi ʻē aʻe.
Hoʻohana 3: Nā lāʻau antitumor.No ka mālama ʻana i ka maʻi maʻi umauma metastatic a me ka maʻi maʻi ovarian metastatic.Nā lāʻau lāʻau anti-tumor ākea ākea no ka mālama ʻana i ka maʻi maʻi ovarian, ka maʻi maʻi umauma a me nā maʻi ʻē aʻe.
Hoʻohana i ka 4: ʻO ka lāʻau anti-tumor maikaʻi;hoʻopaʻa i ka ʻāpana N-terminal o β-tubulin, hoʻoikaika i nā microtubule paʻa loa, kūʻē i ka depolymerization, pale i ka mahele cell maʻamau a me nā pahele i ka pae G2/M o ka pōʻai cell.
E hoʻohana i ka 5: He lāʻau anti-microtubule, e kāohi ana i ka depolymerization ma o ka hoʻolaha ʻana i ka polymerization tubulin, mālama i ka paʻa o ka tubulin, a me ka pale ʻana i ka mitosis cell.