, Kina Paclitaxel 33069-62-4 Anti-tumor Botanical Medicine for Ovarian Cancer, Breast Cancer hale hana a me nā mea hana |Gentolex
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Paclitaxel 33069-62-4 Anti-tumor Botanical Medicine for Ovarian Cancer, Breast Cancer

ʻO ka wehewehe pōkole:

Kahi hehee: 213 °C

Punila hoʻolapalapa: 774.66°C (manaʻo koʻikoʻi)

Ka hoʻololi kikoʻī: D20 -49°(methanol)

Mānoanoa: 1.0352 (manaʻo koʻikoʻi)

Kaila uila: 9°C

Nā kūlana mālama: 2-8°C

ʻAno: pauka

Ka helu ʻana o ka ʻakika: 11.90±0.20(Wānana ʻia)

Kala: Keʻokeʻo


Huahana Huahana

Huahana Huahana

Huahana Huahana

Inoa Paclitaxel
Helu CAS 33069-62-4
ʻAno molekala C47H51NO14
Kaumaha molekula 853.92
Helu EINECS 608-826-9
Lae paila 774.66°C(Wanamua)
ʻO ka mānoanoa 0.200
Kūlana mālama Hoʻopaʻa ʻia i kahi maloʻo, E mālama i loko o ka pahu hau, 2-8 ° C
Puka Pauda
kalakala Keʻokeʻo
Hoʻopili ʻeke PE + ʻeke Aluminum

Nā huaʻōlelo like

Paclitaxel HCL;Paclitaxel(maoli maoli);Paclitaxelx;N-BENZYL-BETA-PHENYLISOSERINE ESTER;PACLITAXEL, TAXUS BREVIFOLIA;PACLITAXEL, TAXUS SPECIES;PACLITAXOL;PACLITAXEL

Ka hopena lāʻau lapaʻau

wehewehe

ʻO Paclitaxel kahi monomeric diterpenoid i unuhi ʻia mai ka ʻili o ka lāʻau maoli ʻo Taxus lāʻau.Ua hōʻike ʻia ka ʻimi ʻana i ka isotope e pili wale ana ka paclitaxel i nā microtubules polymerized a ʻaʻole i pane me nā dimer tubulin unpolymerized.Ma hope o ka ʻike ʻia ʻana o nā cell i ka paclitaxel, e hōʻiliʻili ʻia ka nui o nā microtubules i loko o nā pūnaewele.ʻO ka hōʻiliʻili ʻana o kēia mau microtubules e hoʻopilikia i nā hana like ʻole o nā cell, ʻoi aku ka paʻa o ka māhele cell i ka mitotic phase a poloka i ka mahele maʻamau o nā cell.Ma o Ⅱ-Ⅲ noiʻi lapaʻau, kūpono ka paclitaxel no ka maʻi maʻi ovarian a me ka maʻi kanesa o ka umauma, a loaʻa pū kekahi hopena curative i ka maʻi kanesa, colorectal cancer, melanoma, poʻo a me ka ʻāʻī maʻi, lymphoma a me ka lolo lolo.

 

Nā hōʻailona

He hopena maikaʻi ia i ka mālama ʻana i ka maʻi maʻi ovarian a me ka platinum a me nā maʻi maʻi ovarian refractory a me ka maʻi maʻi umauma.ʻO ka maʻi maʻi, ka maʻi maʻi ʻōpū o luna, ka maʻi maʻi ʻaʻai liʻiliʻi a me ka maʻi ʻaʻaʻa ʻole liʻiliʻi he manaʻo maikaʻi.

 

Hoʻohana

E hoʻohana i ka 1: Nā hua lāʻau anti-tumor ākea ākea no ka maʻi maʻi ovarian, ka maʻi maʻi umauma, etc.

E hoʻohana i ka 2: nā lāʻau lapaʻau anti-tumor ākea ākea no ka mālama ʻana i ka maʻi maʻi ovarian, ka maʻi maʻi umauma a me nā maʻi ʻē aʻe.

Hoʻohana 3: Nā lāʻau antitumor.No ka mālama ʻana i ka maʻi maʻi umauma metastatic a me ka maʻi maʻi ovarian metastatic.Nā lāʻau lāʻau anti-tumor ākea ākea no ka mālama ʻana i ka maʻi maʻi ovarian, ka maʻi maʻi umauma a me nā maʻi ʻē aʻe.

Hoʻohana i ka 4: ʻO ka lāʻau anti-tumor maikaʻi;hoʻopaʻa i ka ʻāpana N-terminal o β-tubulin, hoʻoikaika i nā microtubule paʻa loa, kūʻē i ka depolymerization, pale i ka mahele cell maʻamau a me nā pahele i ka pae G2/M o ka pōʻai cell.

E hoʻohana i ka 5: He lāʻau anti-microtubule, e kāohi ana i ka depolymerization ma o ka hoʻolaha ʻana i ka polymerization tubulin, mālama i ka paʻa o ka tubulin, a me ka pale ʻana i ka mitosis cell.

 

 


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