| inoa | Tirzepatide Injection Powder |
| Maemae | 99% |
| Ka nana aku | Pauda Lyophilized Keʻokeʻo |
| Hooponopono | ʻAiʻi ma lalo o ke kino |
| Nui | 10mg, 15mg, 20mg, 30mg, 60mg |
| Wai | 3.0% |
| Nā pōmaikaʻi | Lapaʻau ʻana i ka maʻi maʻi maʻi, ke kaumaha |
Tirzepatide Lyophilized Pahu (60 mg)
ʻO Tirzepatide (LY3298176) ka mea mua ʻelua-acting agonist e kuhikuhi ana i ka GIP (glucose-dependent insulinotropic polypeptide) a me GLP-1 (glucagon-like peptide-1). Ua loaʻa iā ia ka ʻae ʻana o US FDA i Mei 2022 no ka mālama ʻana i ka maʻi maʻi type 2 (T2DM) ma ke ʻano he mea hoʻohui i ka meaʻai a me ka hoʻoikaika kino.
Hāʻawi ʻia kēia huahana ma ke ʻano he 60mg lyophilized (freeze-dried) sterile pauka i loko o nā hue, pono e hoʻohui hou ʻia me ka wai bacteriostatic ma mua o ka lawelawe ʻana. Hoʻohālikelike ʻia me ka GLP-1 receptor agonists e like me semaglutide a i ʻole dulaglutide, hōʻike ʻo tirzepatide i ka maikaʻi o ka hoʻomaikaʻi ʻana i ka hoʻoponopono glucose koko, hoʻonui i ka ʻike insulin, a me ke kākoʻo ʻana i ke kaumaha nui. Hāʻawi ʻia kēia mau pōmaikaʻi i kāna ʻano hana synergistic dual-receptor o ka hana.
Nā Pōmaikaʻi Nui
Hoʻoponopono Glycemic
Hoʻoponopono kaumaha
Ola maʻi puʻuwai
Hoʻohana a me ka hoʻohana ʻana
ʻAno maʻi diabetes 2
Obesity / Kaumaha
Hoʻohālikelike ʻia i ka Dosage
| Hōʻike | Hoʻomaka ʻana | Ka Papa Hoo | ʻAha maʻamau | ʻO ka nui loa | Ka pinepine |
|---|---|---|---|---|---|
| ʻAno maʻi diabetes 2 | 2.5 mg i kēlā me kēia pule | E hoʻonui i kēlā me kēia 4 pule (→ 5 → 7.5 → 10 → 12.5 → 15 → 20 → 30 → 45 → 60) | 10-30 mg i kēlā me kēia pule | 60 mg i kēlā me kēia pule | Hoʻokahi pule i kēlā me kēia pule |
| Obesity / Weight Loss | 2.5 mg i kēlā me kēia pule | Hoʻonui ma muli o ka hoʻomanawanui (2.5 → 5 → 7.5 → 10 → 12.5 → 15 → 20 → 30 → 45 → 60) | 30-60 mg i kēlā me kēia pule | 60 mg i kēlā me kēia pule | Hoʻokahi pule i kēlā me kēia pule |
Nānā:E hōʻoia i kēlā me kēia maʻi mua e ʻae maikaʻi ʻia ma mua o ka piʻi ʻana.
ʻO nā hopena ʻino paha
Pharmacokinetics
Hōʻuluʻulu manaʻo
ʻO Tirzepatide 60 mg lyophilized pauka e hōʻike ana i ka holomua therapeutic o ka hanauna e hiki mai ana, e hui pū ana i ka mana glycemic ikaika me ka maikaʻi o ka pohō kaumaha a me ka pale cardiovascular.
Me ka papa kuhikuhi titration lohi (2.5 mg → a hiki i 60 mg), hiki iā ia ke hoʻonui i ka hoʻomanawanui a me ka maʻalahi no ka mālama pilikino. ʻO kāna hoʻokele hoʻokahi pule i hoʻomaikaʻi i ka pili ʻana, e lilo ia i koho hou a maikaʻi hoʻi no ka mālama ʻana i ka maʻi maʻi type 2 a me ka momona i nā hoʻonohonoho hoʻokolohua holomua a me ka noiʻi.